Elagolix Racemic Mixture

It is an impurity present in Elagolix, Elagolix is a gonadotropin-releasing hormone receptor antagonist that inhibits endogenous GnRH, By administration of elagolix shows results in dose-dependent suppression of luteinizing hormone and follicle-stimulating hormone, which leads to decreased blood concentrations of the ovarian sex hormones, estradiol, and progesterone, which is used to treat moderate to severe pain in endometriosis.

Additional information on Elagolix Racemic Mixture

Catalogue No.

VE006430

CAS No.

N/A

Molecular Formula

C32H29F5N3NaO5

Molecular Weight

653.57

Parent drug

Elagolix

IUPAC Name

Sodium (R, S)-4-((2-(5-(2-fluoro-3-methoxyphenyl)-3-(2-fluoro-6-(trifluoromethyl)benzyl)-4-methyl-2, 6-dioxo-2, 3-dihydropyrimidin-1(6H)-yl)-1-phenylethyl)amino)butanoate

Synonyms

N/A

References

Archer, D. F., Soliman, A. M., Agarwal, S. K., & Taylor, H. S. (2020). Elagolix in the treatment of endometriosis: impact beyond pain symptoms. Therapeutic Advances in Reproductive Health, 14, 263349412096451. https://doi.org/10.1177/2633494120964517 ‌Lamb, Yvette N. “Elagolix: First Global Approval.” Drugs, vol. 78, no. 14, Sept. 2018, pp. 1501–8, https://doi.org/10.1007/s40265-018-0977-4. ‌

Status

Under Development

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Elagolix Racemic Mixture

Elagolix Racemic Mixture
Catalogue No.

VE006430

CAS No.

N/A

Molecular Formula

C32H29F5N3NaO5

Molecular Weight

653.57

Parent drug

Elagolix

IUPAC Name

Sodium (R, S)-4-((2-(5-(2-fluoro-3-methoxyphenyl)-3-(2-fluoro-6-(trifluoromethyl)benzyl)-4-methyl-2, 6-dioxo-2, 3-dihydropyrimidin-1(6H)-yl)-1-phenylethyl)amino)butanoate

Synonyms

N/A

References

Archer, D. F., Soliman, A. M., Agarwal, S. K., & Taylor, H. S. (2020). Elagolix in the treatment of endometriosis: impact beyond pain symptoms. Therapeutic Advances in Reproductive Health, 14, 263349412096451. https://doi.org/10.1177/2633494120964517 ‌Lamb, Yvette N. “Elagolix: First Global Approval.” Drugs, vol. 78, no. 14, Sept. 2018, pp. 1501–8, https://doi.org/10.1007/s40265-018-0977-4. ‌

Status

Under Development

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Elagolix Racemic Mixture

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